Lately reported that A-893, a benzoxazinone derivative, specifically inhibits SMYD2 enzyme activity (IC50, 2.eight nM).
Lately reported that A-893, a benzoxazinone derivative, specifically inhibits SMYD2 enzyme activity (IC50, 2.eight nM). This inhibitor clearly suppressed p53K370 methylation mediated by SMYD2 in lung carcinoma A549 cells. For…